苯噻啶苹果酸盐 ,≥98.5%

Pizotifen Malate
别名:
Cas号: 5189-11-7 物化性质:
分子式: C23H27NO5S 熔点:
分子量: 429.529185533524 沸点:
EINECS编号: 225-970-4 密度:
MDL号: 储存条件: 2-8℃

物理性状及指标:

外观:……………………白色或类白色结晶性粉末

熔点:……………………365-366.8 °C (dec.)

溶解性:…………………溶于水(3 mg/ml)和DMSO (30 mg/ml)

干燥失重:………………≤0.5%

含量:……………………98.5%~101.5%

IC50:……………………半数致死剂量 (LD50) 经口 - 大鼠 - 410 mg/kg

用途及描述:科研试剂,广泛应用于分子生物学,药理学等科研方面。苯噻啶是一种血清素拮抗剂,主要作用于5-HT1、5-HT2A和5HT2C受体,还具有抗组胺剂活性。可用于预防血管性头痛包括偏头痛和丛集性头痛

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苯噻啶苹果酸盐
malic acid, compound with 4-(9,10-dihydro-4H-benzo[4,5]cyclohepta[1,2-b]thien-4-ylidene)-1-methylpiperidine (1:1);Pizotifen Malate;PIZOTIFEN MALATE BP GRADE B.P.98;Pizotyline malate;4-(4,5-dihydrobenzo[1,2]cyclohepta[3,4-b]thiophen-10-ylidene)-1-methylpiperidine,2-hydroxybutanedioic acid;Litec malate;Mosegor;Pizotifen hydrogen malate;Sandomigran;Sandomigran malate;Sandomigran,pizotyline;Sandomygran malate;Sanomtgran;Butanedioicacid, hydroxy-, compd. with4-(9,10-dihydro-4H-benzo[4,5]cyclohepta[1,2-b]thien-4-ylidene)-1-methylpiperidine(1:1) (9CI);Malic acid, compd. with 4-(9,10-dihydro-4H-benzo[4,5]cyclohepta[1,2-b]thien-4-ylidene)-1-methylpiperidine(1:1) (8CI);Malic acid, compd. with4-(9,10-dihydro-4H-benzo[4,5]cyclohepta[1,2-b]thien-4-ylidene)-1-methylpiperidine(7CI);4H-Benzo[4,5]cyclohepta[1,2-b]thiophene, 9,10-dihydro-4-(1-methyl-4-piperidylidene)-,malate (1:1) (8CI);4H-Benzo[4,5]cyclohepta[1,2-b]thiophene, piperidine deriv.;Piperidine,4-(9,10-dihydro-4H-benzo[4,5]cyclohepta[1,2-b]thien-4-ylidene)-1-methyl-,hydroxybutanedioate (1:1) (9CI);Piperidine, 4-(9,10-dihydro-4H-benzo[4,5]cyclohepta[1,2-b]thien-4-ylidene)-1-methyl-,malate (1:1) (8CI);4-(9,10-Dihydro-4H-benzo[4,5]cyclohepta[1,2-b]thien-4-ylidene)-1-methylpiperidiniumhydrogen malate;Pizotifen malate;Sanmigran;Sanomigran;9,10-Dihydro-4-(1-methylpiperidin-4-ylidene)-4H-benzo[4,5]cyclohepta[1,2-b]thiophene malate (1:1)